激酶抑制劑 kinase inhibitor
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激酶 (kinase) 具有調節細胞之間訊號傳遞的生理功能。酵素激酶所建構出的網絡系統 (kinase network),參與體內所有的生理反應。在基礎實驗與新藥開發等的科研領域中,透過干擾激酶的作用,探究小分子標靶對於生理功能的重要性,開發出最具生理意義的重要小分子。
這篇部落格詳細記錄重要的酵素激酶抑制劑,讓研究者有更多更好的抑制劑選擇,並進一步了解探索激酶在生理功能上的運轉。
EGFR/ErbB/HER Family | |
Afatinib | 11492 |
AZD 9291 | 16237 |
Erlotinib | 10483 |
Gefitinib | 13166 |
Lapatinib | 11493 |
MEK | |
AZD 6244 | 11599 |
BIX02189 | 16999 |
PD 0325901 | 13034 |
Trametinib | 16292 |
U-0126 | 70970 |
JNK | |
Bentamapimod | 21482 |
JNK Inhibitor V | 17542 |
JNK Inhibitor VIII | 15946 |
JNK Inhibitor XVI | 18096 |
SP 600125 | 10010466 |
IGF-1R | |
AG-1024 | 14833 |
BMS 754807 | 17505 |
Linsitinib | 17708 |
NVP-AEW541 (hydrochloride) | 13641 |
Picropodophyllotoxin | 17329 |
p38 MAPK | |
Doramapimod | 10460 |
PD 169316 | 10006727 |
SB 202190 | 10010399 |
SB 203580 | 13067 |
VX-745 | 18075 |
JAK Family | |
Baricitinib | 16707 |
CP 690,550 | 11598 |
Filgotinib | 17669 |
Lestaurtinib | 12094 |
Ruxolitinib | 11609 |
PI3K | |
BYL719 | 16986 |
CAL-101 | 15279 |
LY294002 | 70920 |
TGR-1202 | 32877 |
Wortmannin | 10010591 |
PKB/Akt | |
A-443654 | 16499 |
Akt Inhibitor VIII | 14870 |
AZD 5363 | 15406 |
GDC-0068 | 18412 |
ML-9 | 10010236 |
ERK | |
FR180204 | 15544 |
GDC-0994 | 21107 |
SCH 772984 | 19166 |
Ulixertinib (hydrochloride) | 18298 |
XMD8-92 | 19173 |
mTOR | |
AZD 8055 | 16978 |
PP242 | 13643 |
Rapamycin | 13346 |
Torin 1 | 10997 |
Torin 2 | 14185 |
PDPK1/PDK1 | |
BX-795 | 14932 |
BX-912 | 14708 |
GSK2334470 | 18095 |
KT 5720 | 10011011 |
UCN-01 | 18130 |
PKC | |
Calphostin C | 15383 |
Gö 6976 | 13310 |
Gö 6983 | 13311 |
LY333531 (hydrochloride) | 13964 |
Staurosporine | 81590 |
IKKs | |
BMS 345541 (hydrochloride) | 16667 |
IKK-16 (hydrochloride) | 13313 |
IKK2 Inhibitor VI | 17276 |
IMD 0354 | 17290 |
TPCA-1 | 15115 |
GSK3 | |
1-Azakenpaullone | 16733 |
BIO | 13123 |
CHIR99021 | 13122 |
SB-216763 | 10010246 |
TWS119 | 10011251 |
Plks | |
BI-2536 | 17385 |
BI-6727 | 18193 |
GSK461364 | 18099 |
ON-01910 (sodium salt) | 15553 |
TAK-960 | 17701 |
Src | |
CGP 77675 (hydrate) | 21089 |
PP1 (Src Inhibitor) | 14244 |
PP2 | 13198 |
Saracatinib | 11497 |
SU6656 | 13338 |
Abl Family & Bcr-Abl | |
Bosutinib | 12030 |
Dasatinib | 11498 |
Imatinib (mesylate) | 13139 |
Nilotinib | 10010422 |
Ponatinib | 11494 |
CDKs | |
Dinaciclib | 14707 |
Flavopiridol (hydrochloride) | 10009197 |
PD 0322991 (hydrochloride) | 16273 |
Ro 3306 | 15149 |
Senexin B | 28459 |
CSF1R/Fms | |
BLZ-945 | 19626 |
Edicotinib | 33347 |
Ki20227 | 22258 |
Pexidartinib | 18271 |
PLX5622 | 28927 |
ALK (Anaplastic Lymphoma Kinase) | |
AP26113 | 19778 |
Ceritinib | 19374 |
CH5424802 | 18516 |
PF-06463922 | 18371 |
TAE684 | 17670 |
Chk1/2 | |
AZD 7762 | 11491 |
CCT241533 (hydrochloride) | 19178 |
LY2603618 | 20351 |
LY2606368 | 21490 |
PF-477736 | 17859 |
DNA-PK | |
CC-115 | 19420 |
Ku-0060648 | 15344 |
NU 7026 | 13308 |
NU 7441 | 14881 |
PI-103 | 10009209 |
FGFR Family | |
AZD 4547 | 13111 |
BGJ398 | 19157 |
JNJ-42756493 | 21813 |
PD 173074 | 13032 |
TAS 120 | 21136 |
Aurora | |
AMG 900 | 19176 |
MLN8237 | 13602 |
PF-03814735 | 15015 |
Phthalazionone pyrazole | 10735 |
ZM 447439 | 13601 |
c-Met | |
(R)-Crizotinib | 12087 |
Golvatinib | 22143 |
INCB 28060 | 20056 |
SU11274 | 14861 |
Tivantinib | 17135 |
FLT3 | |
FLT3 Inhibitor III | 21193 |
Gilteritinib | 21503 |
Pacritinib | 16709 |
Quizartinib | 17986 |
UNC2025 | 16613 |
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發佈時間 May 02, 2022
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